Confirmation of HTS candidates by FP competition assay.
2015-09-14T02:46:08Z (GMT) by
A and B. 5 nM F12-ATP and 200 nM GST-HEPN were titrated with the hits to confirm their binding to GST-HEPN. C. Affinities of the compounds for HEPN were estimated from the competition assays and summarized along with their chemical structures.