10.1371/journal.pntd.0004617.t003
Diego Benítez
Diego
Benítez
Andrea Medeiros
Andrea
Medeiros
Lucía Fiestas
Lucía
Fiestas
Esteban A. Panozzo-Zenere
Esteban A.
Panozzo-Zenere
Franziska Maiwald
Franziska
Maiwald
Kyriakos C. Prousis
Kyriakos C.
Prousis
Marina Roussaki
Marina
Roussaki
Theodora Calogeropoulou
Theodora
Calogeropoulou
Anastasia Detsi
Anastasia
Detsi
Timo Jaeger
Timo
Jaeger
Jonas Šarlauskas
Jonas
Šarlauskas
Lucíja Peterlin Mašič
Lucíja Peterlin
Mašič
Conrad Kunick
Conrad
Kunick
Guillermo R. Labadie
Guillermo R.
Labadie
Leopold Flohé
Leopold
Flohé
Marcelo A. Comini
Marcelo
A. Comini
Compounds enhancing tritryp trypanothione synthetase (TryS) activity.
Public Library of Science
2016
broad-range TryS inhibitors
screening
compound
drug target candidate
trypanothione
infective Trypanosoma brucei
Novel Chemical Scaffolds Inhibiting Trypanothione Synthetase
MOL
novel chemical entities
Several novel chemical scaffolds
EC 50
tri-tryp TryS inhibitors
Leishmania infantum promastigotes
Pathogenic Trypanosomatids Background
thiol-dependent redox metabolism
trypanosomatid
2016-04-12 23:01:17
Dataset
https://plos.figshare.com/articles/dataset/Compounds_enhancing_tritryp_trypanothione_synthetase_TryS_activity_/3951855
<p>Compounds enhancing tritryp trypanothione synthetase (TryS) activity.</p>